7-PET: Difference between revisions

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'''7-PET''' is a potent [[analgesic]] drug, several thousand times stronger than [[morphine]] by weight. It is related to the more well-known [[oripavine]] derivative opioid [[etorphine]], which is used as a very potent [[veterinary]] painkiller and [[anesthetic]] medication, used primarily for the sedation of large animals such as elephants, giraffes and rhinos. 7-PET is around the same potency as etorphine as a [[mu opioid receptor|μ]] [[agonist]].<ref>Feinberg AP, Creese I, Snyder SH. The opiate receptor: a model explaining structure-activity relationships of opiate agonists and antagonists. ''Proceedings of the National Academy of Sciences U S A''. 1976 Nov;73(11):4215-9.</ref><ref>Bentley KW, Lewis JW. Agonist and Antagonist Actions of Narcotic Analgesic Drugs. pp 7-16. University Park Press, Baltimore. (1973)</ref>
'''7-PET''' is a potent [[analgesic]] drug, several thousand times stronger than [[morphine]] by weight. It is related to the more well-known [[oripavine]] derivative opioid [[etorphine]], which is used as a very potent [[veterinary]] painkiller and [[anesthetic]] medication, used primarily for the sedation of large animals such as elephants, giraffes and rhinos. 7-PET is around the same potency as etorphine as a [[mu opioid receptor|μ]] [[agonist]].<ref>Feinberg AP, Creese I, Snyder SH. The opiate receptor: a model explaining structure-activity relationships of opiate agonists and antagonists. ''Proceedings of the National Academy of Sciences U S A''. 1976 Nov;73(11):4215-9.</ref><ref>Bentley KW, Lewis JW. Agonist and Antagonist Actions of Narcotic Analgesic Drugs. pp 7-16. University Park Press, Baltimore. (1973)</ref>

Latest revision as of 19:07, 8 August 2012

7-PET
File:7-PET.svg
Identifiers
E number{{#property:P628}}
ECHA InfoCard{{#property:P2566}}Lua error in Module:EditAtWikidata at line 36: attempt to index field 'wikibase' (a nil value).
Chemical and physical data
FormulaC31H37NO4
Molar mass487.64 g/mol


7-PET is a potent analgesic drug, several thousand times stronger than morphine by weight. It is related to the more well-known oripavine derivative opioid etorphine, which is used as a very potent veterinary painkiller and anesthetic medication, used primarily for the sedation of large animals such as elephants, giraffes and rhinos. 7-PET is around the same potency as etorphine as a μ agonist.[1][2]

Unlike etorphine however, 7-PET is not an illegal drug, and is not controlled under the UN drug conventions, but it might still be considered to be a controlled substance analogue of etorphine on the grounds of its related chemical structure in some jurisdictions such as the USA, Canada, Australia and New Zealand.

References

  1. ↑ Feinberg AP, Creese I, Snyder SH. The opiate receptor: a model explaining structure-activity relationships of opiate agonists and antagonists. Proceedings of the National Academy of Sciences U S A. 1976 Nov;73(11):4215-9.
  2. ↑ Bentley KW, Lewis JW. Agonist and Antagonist Actions of Narcotic Analgesic Drugs. pp 7-16. University Park Press, Baltimore. (1973)

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